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    A matrix-focused structure-activity and binding site flexibility study of quinolinol inhibitors of botulinum neurotoxin serotype A 

    Harrell, William A. Jr.; Vieira, Rebecca C.; Ensel, Susan M.; Montgomery, Vicki; Guernieri, Rebecca; Eccard, Vanessa S.; Campbell, Yvette; Roxas-Duncan, Virginia; Cardellina, John H. II; Webb, Robert P.; Smith, Leonard A. (Bioorganic & Medicinal Chemistry Letters, 2017-02-01)
    Our initial discovery of 8-hydroxyquinoline inhibitors of BoNT/A and separation/testing of enantiomers of one of the more active leads indicated considerable flexibility in the binding site. We designed a limited study to ...


    Stevenson University Library
    1525 Greenspring Valley Road
    Stevenson, MD 21153

    Website: http://stevensonlibrary.org

    Contact information:
    Elizabeth Fields
    efields2@stevenson.edu
    http://stevenson.libguides.com/sse


    If you wish to submit a copyright complaint or withdrawal request, please email mdsoar-help@umd.edu.

     

     

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    AuthorCampbell, Yvette (1)Cardellina, John H. II (1)Eccard, Vanessa S. (1)Ensel, Susan M. (1)Guernieri, Rebecca (1)Harrell, William A. Jr. (1)Montgomery, Vicki (1)Roxas-Duncan, Virginia (1)Smith, Leonard A. (1)Vieira, Rebecca C. (1)... View MoreSubject
    Animals (1)
    Binding Sites (1)Botulinum Toxins, Type A--antagonists & inhibitors (1)Botulinum Toxins, Type A--metabolism (1)Hydroxyquinolines--chemistry (1)Hydroxyquinolines--metabolism (1)Hydroxyquinolines--toxicity (1)Inhibitory Concentration 50 (1)Mice (1)Phrenic Nerve--drug effects (1)... View MoreDate Issued2017 (1)Has File(s)No (1)


    Stevenson University Library
    1525 Greenspring Valley Road
    Stevenson, MD 21153

    Website: http://stevensonlibrary.org

    Contact information:
    Elizabeth Fields
    efields2@stevenson.edu
    http://stevenson.libguides.com/sse


    If you wish to submit a copyright complaint or withdrawal request, please email mdsoar-help@umd.edu.